Kazia reports 52% preclinical tumor-burden reduction for paxalisib in resistant colorectal cancer

  • Kazia reported paxalisib reduced tumor burden in preclinical MSS/pMMR colorectal cancer.
  • 52% tumor-burden reduction occurred with paxalisib monotherapy, with p=0.035.
  • Kazia plans five-arm Phase 2 enrollment during the first quarter of 2027.

Kazia Therapeutics said paxalisib reduced tumor burden by 52% in a preclinical model of microsatellite stable, proficient mismatch repair colorectal cancer, with statistical significance of p=0.035. Adding paxalisib to pembrolizumab reduced tumor volume by a further 50% versus pembrolizumab alone in a separate study, with p=0.022. Treatments were well tolerated without evidence of treatment-related toxicity. Kazia is developing biomarker analyses and plans to begin a five-arm Phase 2 trial in pre-treated MSS/pMMR metastatic colorectal cancer during the first quarter of 2027, comparing two paxalisib doses, combinations with pembrolizumab with or without biologic, and standard of care.

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